Chroman-4-ol → HCID 58900201, compound

Participants

Reaction Steps

The title compound was prepared as a white solid (58 mg, 53% yield for 2 steps) from 1,1-dimethylethyl 6-[(dimethylamino)carbonyl]-4-hydroxy-2-methyl-1H-benzimidazole-1-carboxylate (100 mg, 0.313 mmol, STEP 2 in Example 9) and 3,4-dihydro-2H-chromen-4-ol (141 mg, 0.939 mmol) by the same manner in STEP 3-2 of Example 9:

Provenance & Evidence