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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2245519Generated: November 2, 2026

4-t-Butylbenzenesulfonyl chloride → N-{4-[(5-{[(4-tert-Butylphenyl)sulfonyl]amino}-1H-indol-1-yl)methyl]benzoyl}-L-phenylalanine

https://huagongshe.com/reaction/2245519

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-t-Butylbenzenesulfonyl chlorideHCID 139882—
Reactantethyl N-{4-[(5-amino-1H-indol-1-yl)methyl]benzoyl}phenylalaninateHCID 68548160—
ProductN-{4-[(5-{[(4-tert-Butylphenyl)sulfonyl]amino}-1H-indol-1-yl)methyl]benzoyl}-L-phenylalanineHCID 16113985—

Reaction Steps

The title compound was prepared from ethyl N-{4-[(5-amino-1H-indol-1-yl)methyl]benzoyl}phenylalaninate and 4-tert-butylphenyl sulfonyl chloride following the procedure of Example 10: MS (ESI) m/z 610; MS (ESI) m/z 608.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07683091B2
Source datasetuspto-grants-2010_03
ORD IDord-b0183e3bac29402892016aa3d55b43f9
Source noteuspto-grants-2010_03