Benzoyl isocyanate → HCID 56982097, compound

HRID 225150Notes

Reaction equation

[NH2:1][CH:2]1[CH2:7][CH2:6][N:5]([CH2:8][CH:9]([CH:11]2[O:16][C:15]3[CH:17]=[CH:18][C:19]([O:21][CH3:22])=[CH:20][C:14]=3[O:13][CH2:12]2)[OH:10])[CH2:4][CH2:3]1.[C:23]([N:31]=[C:32]=[O:33])(=[O:30])[C:24]1[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=1>>[C:23]([NH:31][C:32]([NH:1][CH:2]1[CH2:7][CH2:6][N:5]([CH2:8][CH:9]([CH:11]2[O:16][C:15]3[CH:17]=[CH:18][C:19]([O:21][CH3:22])=[CH:20][C:14]=3[O:13][CH2:12]2)[OH:10])[CH2:4][CH2:3]1)=[O:33])(=[O:30])[C:24]1[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=1

Participants

Reactant 2

HCID 78210Benzoyl isocyanate

HCID 57158659HCID 57158659, compound

Product 1

HCID 56982097HCID 56982097, compound

Procedure

Using the procedure of Example 4 erythro 4-amino-1-[2-(6-methoxy-1,4-benzodioxan-2-yl)-2-hydroxyethyl]piperidine may be reacted with benzoyl isocyanate to give the title compound.

Sources & evidence

ORD record: ord-6d17f97ac32749cbbcfd6b76e388417e
Source dataset: uspto-grants-1980_11
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US04235915

Reaction notes

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