HCID 10016688, compound → HCID 9981705, compound

HRID 2255313Notes

Reaction equation

HRID 2255313 reaction equation
[NH2:1][C:2]1[CH:16]=[CH:15][CH:14]=[CH:13][C:3]=1[O:4][CH2:5][CH2:6][CH2:7][C:8]([O:10]CC)=[O:9].[CH:17]1([N:23]2[C:31]3[C:26](=[CH:27][C:28](/[C:32](/[CH3:37])=[CH:33]/[C:34](O)=[O:35])=[CH:29][CH:30]=3)[CH:25]=[CH:24]2)[CH2:22][CH2:21][CH2:20][CH2:19][CH2:18]1>>[CH:17]1([N:23]2[C:31]3[C:26](=[CH:27][C:28](/[C:32](/[CH3:37])=[CH:33]/[C:34]([NH:1][C:2]4[CH:16]=[CH:15][CH:14]=[CH:13][C:3]=4[O:4][CH2:5][CH2:6][CH2:7][C:8]([OH:10])=[O:9])=[O:35])=[CH:29][CH:30]=3)[CH:25]=[CH:24]2)[CH2:18][CH2:19][CH2:20][CH2:21][CH2:22]1

Participants

3

Reactant 2

HCID 10016688HCID 10016688, compoundHCID 11816929Ethyl 4-(2-aminophenoxy)butanoate

Product 1

HCID 9981705HCID 9981705, compound

Procedure

0.22 g of compound 24 was obtained in a similar manner to those described in the Examples 1 to 2 using 0.47 g of ethyl 4-(2-aminophenoxy)butyrate and 0.30 g of 3-(1-cyclohexylindol-5-yl)isocrotonic acid obtained according to the procedures described in the Reference Examples 1-4.

Workup

  1. customobtained

Sources & evidence

ORD record
ord-72e2d7dd7d564317aeacfbdd8bf1aa19
Source dataset
uspto-grants-1993_08
Patent number
US05239083

Reaction notes

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