HCID 10472882, compound → HCID 10414473, compound

HRID 2255328Notes

Reaction equation

HRID 2255328 reaction equation
[NH2:1][C:2]1[CH:16]=[CH:15][CH:14]=[CH:13][C:3]=1[O:4][CH2:5][CH2:6][CH2:7][C:8]([O:10]CC)=[O:9].[CH2:17]([CH:21]([N:28]1[C:36]2[C:31](=[CH:32][C:33](/[C:37](/[CH3:42])=[CH:38]/[C:39](O)=[O:40])=[CH:34][CH:35]=2)[CH:30]=[CH:29]1)[C:22]1[CH:27]=[CH:26][CH:25]=[CH:24][CH:23]=1)[CH2:18][CH2:19][CH3:20]>>[CH2:17]([CH:21]([N:28]1[C:36]2[C:31](=[CH:32][C:33](/[C:37](/[CH3:42])=[CH:38]/[C:39]([NH:1][C:2]3[CH:16]=[CH:15][CH:14]=[CH:13][C:3]=3[O:4][CH2:5][CH2:6][CH2:7][C:8]([OH:10])=[O:9])=[O:40])=[CH:34][CH:35]=2)[CH:30]=[CH:29]1)[C:22]1[CH:23]=[CH:24][CH:25]=[CH:26][CH:27]=1)[CH2:18][CH2:19][CH3:20]

Participants

3

Reactant 2

HCID 10472882HCID 10472882, compoundHCID 11816929Ethyl 4-(2-aminophenoxy)butanoate

Product 1

HCID 10414473HCID 10414473, compound

Procedure

0.61 g of compound 42 was obtained in a similar manner to those described in the Examples 1 and 2 using 1.28 g of ethyl 4-(2-aminophenoxy)butyrate and 1.0 g of 3-[1-(α-butylbenzyl)indol-5-yl]isocrotonic acid obtained according to the procedures described in the Reference Examples 1-4.

Workup

  1. customobtained

Sources & evidence

ORD record
ord-67cc2be934784125a078c2d7505f69f0
Source dataset
uspto-grants-1993_08
Patent number
US05239083

Reaction notes

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