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3-Fluoro-5-(trifluoromethyl)benzeneboronic acid → HCID 57755059、化合物
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 3-Fluoro-5-(trifluoromethyl)benzeneboronic acid | HCID 2783192 | — |
| 反応物 | 2-(3'-Fluoro-5-hydroxy-5'-trifluoromethyl-biphenyl-3-yl)-4-methyl-pentanoic acid methyl ester | HCID 57755035 | — |
| 生成物 | HCID 57755059 | HCID 57755059 | 73% |
反応手順
The title compound was prepared in 73% yield from 2-(3′-fluoro-5-hydroxy-5′-trifluoromethyl-biphenyl-3-yl)-4-methyl-pentanoic acid methyl ester (prepared in Example B) and 3-fluoro-5-trifluoromethylbenzene boronic acid under the conditions described in Example 15, step (g).
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US07557244B2 |
| 出典データセット | uspto-grants-2009_07 |
| ORD ID | ord-81b96f410ef448aba81eeeca9fc95dfe |
| 出典メモ | uspto-grants-2009_07 |