HCID 57807712, compound → HCID 57807461, compound

Participants

Role	Name	HCID	Charge
Reactant	HCID 57807712	HCID 57807712	—
Reactant	(R)-2-(4-amino-3-chloro-5-trifluoromethyl-phenyl)-1-carboxy-ethyl 4-(2-oxo-1,2,4,5-tetrahydro-1,3-benzodiazepin-3-yl)-piperidine-1-carboxylate	HCID 58202073	—
Product	HCID 57807461	HCID 57807461	—

Reaction Steps

Prepared analogously to Example 24 from 500 mg (0.90 mmol) (R)-2-(4-amino-3-chloro-5-trifluoromethyl-phenyl)-1-carboxy-ethyl 4-(2-oxo-1,2,4,5-tetrahydro-1,3-benzodiazepin-3-yl)-piperidine-1-carboxylate (Example 1f) and 341 mg (1.00 mmol) ethyl 3-[1,4′]bipiperidinyl-4-yl-propionate (Example A15b).

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US07858622B2
Source dataset	uspto-grants-2010_12
ORD ID	ord-934458d56d244d7b8b5115d446bbc7e9
Source note	uspto-grants-2010_12