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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2267863Generated: October 31, 2026

4-phenoxy-1H-indole-2-carboxylic acid → 4-Phenoxy-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide

https://huagongshe.com/reaction/2267863

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-phenoxy-1H-indole-2-carboxylic acidHCID 59600239—
Reactant1-(2-(Azepan-1-yl)ethyl)piperidin-4-amine trihydrochlorideHCID 66841393—
Product4-Phenoxy-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amideHCID 59600154—

Reaction Steps

This compound is synthesized analogously to Example 1 from 4-phenoxy-1H-indole-2-carboxylic acid 129 (preparation see below) and amine 5.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07858781B2
Source datasetuspto-grants-2010_12
ORD IDord-0a252805413744608416c9e1886fbdac
Source noteuspto-grants-2010_12