Benzo[C][1,2,5]Oxadiazole-5-Boronic Acid → 4-Benzo[1,2,5]oxadiazol-5-yl-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide

Participants

Role	Name	HCID	Charge
Reactant	Benzo[C][1,2,5]Oxadiazole-5-Boronic Acid	HCID 4672597	—
Reactant	4-Bromo-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide	HCID 59600248	—
Product	4-Benzo[1,2,5]oxadiazol-5-yl-1H-indole-2-carboxylic acid [1-(2-azepan-1-yl-ethyl)-piperidin-4-yl]-amide	HCID 59600240	—

Reaction Steps

This compound is synthesized from compound 194 (see example 156) and benzo[1,2,5]oxadiazol-5-yl-boronic acid analogously to the method described in Example 156.

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US07858781B2
Source dataset	uspto-grants-2010_12
ORD ID	ord-174845084c654813a046a78d1650dafd
Source note	uspto-grants-2010_12