2-Cyanopyridine-5-boronic acid pinacol ester → HCID 178450275, compound

Participants

Reaction Steps

Following general procedure D, tert-butyl trans-4-(6-bromo-3-isobutyrylquinolin-4-ylamino)cyclohexylcarbamate (47 mg, 0.093 mmol) was reacted with 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile (26 mg, 0.200 mmol) to afford the crude product (47 mg) as a yellow solid: ESI MS m/z 514 [C30H35N5O3+H]+.

Provenance & Evidence