HCID 86725183, compound → HCID 86725182, compound

HRID 2276356Notes

Reaction equation

HRID 2276356 reaction equation
[F:1][C:2]1[CH:14]=[CH:13][C:5]2[CH2:6][C@H:7](OC)[B:8]([OH:10])[O:9][C:4]=2[C:3]=1[C:15]([OH:17])=[O:16].[NH2:18][N:19]1[CH:23]=[N:22][N:21]=[C:20]1[SH:24]>>[NH2:18][N:19]1[CH:23]=[N:22][N:21]=[C:20]1[S:24][C@H:7]1[CH2:6][C:5]2[CH:13]=[CH:14][C:2]([F:1])=[C:3]([C:15]([OH:17])=[O:16])[C:4]=2[O:9][B:8]1[OH:10]

Participants

3

Reactant 2

HCID 86725183HCID 86725183, compoundHCID 178514271HCID 178514271, compound

Product 1

HCID 86725182HCID 86725182, compound

Procedure

Compound (20) was prepared from 19G (example 19) following methods described in steps 5 and 6 of example 1 utilizing 4-amino-4H-1,2,4-triazole-3-thiol.

Sources & evidence

ORD record
ord-53c6ffebc21c4c9c838224f23cbe7c98
Source dataset
uspto-grants-2015_09
Patent number
US09132140B2

Reaction notes

Loading…