HCID 86725183, compound → HCID 86725187, compound

HRID 2276359Notes

Reaction equation

HRID 2276359 reaction equation
[F:1][C:2]1[CH:14]=[CH:13][C:5]2[CH2:6][C@H:7](OC)[B:8]([OH:10])[O:9][C:4]=2[C:3]=1[C:15]([OH:17])=[O:16].[CH3:18][N:19]1[CH:23]=[N:22][N:21]=[C:20]1[SH:24]>>[F:1][C:2]1[CH:14]=[CH:13][C:5]2[CH2:6][C@H:7]([S:24][C:20]3[N:19]([CH3:18])[CH:23]=[N:22][N:21]=3)[B:8]([OH:10])[O:9][C:4]=2[C:3]=1[C:15]([OH:17])=[O:16]

Participants

3

Reactant 2

HCID 86725183HCID 86725183, compoundHCID 178481306HCID 178481306, compound

Product 1

HCID 86725187HCID 86725187, compound

Procedure

Compound 24 was prepared from Compound 19G (example 19) following methods described in steps 5 and 6 of Example 1 utilizing 4-methyl-3-mercapto-1,2,4-triazole.

Sources & evidence

ORD record
ord-ece3fdafb2e842169982b712385226e1
Source dataset
uspto-grants-2015_09
Patent number
US09132140B2

Reaction notes

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