HCID 15408835, compound → HCID 86731343, compound

HRID 2277267Notes

Reaction equation

HRID 2277267 reaction equation
[CH2:1]([O:8][C:9]1[CH:14]=[CH:13][C:12]([C:15]2[O:16][C:17]3[CH:23]=[C:22]([OH:24])[CH:21]=[CH:20][C:18]=3[N:19]=2)=[CH:11][C:10]=1[F:25])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.O[CH:27]([CH3:38])[C@@H:28]([NH:30][C:31](=[O:37])[O:32][C:33]([CH3:36])([CH3:35])[CH3:34])[CH3:29]>>[CH2:1]([O:8][C:9]1[CH:14]=[CH:13][C:12]([C:15]2[O:16][C:17]3[CH:23]=[C:22]([O:24][CH:27]([CH3:38])[C@@H:28]([NH:30][C:31](=[O:37])[O:32][C:33]([CH3:36])([CH3:35])[CH3:34])[CH3:29])[CH:21]=[CH:20][C:18]=3[N:19]=2)=[CH:11][C:10]=1[F:25])[C:2]1[CH:3]=[CH:4][CH:5]=[CH:6][CH:7]=1

Participants

3

Reactant 2

HCID 15408835HCID 15408835, compoundHCID 86731344HCID 86731344, compound

Product 1

HCID 86731343HCID 86731343, compound

Procedure

Using 2-(4-(benzyloxy)-3-fluorophenyl)-1,3-benzoxazol-6-ol and tert-butyl ((2S)-3-hydroxybutan-2-yl)carbamate, and in the same manner as in Step C of Example 1, the title compound was obtained.

Sources & evidence

ORD record
ord-8beecf94d686457fb5b1d98a1d0539a6
Source dataset
uspto-grants-2015_09
Patent number
US09133129B2

Reaction notes

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