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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2277406Generated: October 31, 2026

1-Ethyl-3-(3'-dimethylaminopropyl)carbodiimide → N-(4-((7-hydroxy-6-methoxyquinolin-4-yl)oxy)phenyl)-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide

https://huagongshe.com/reaction/2277406

Reaction equation

Participants

RoleNameHCIDCharge
Reactant1-Ethyl-3-(3'-dimethylaminopropyl)carbodiimideHCID 15908—
ReactantHOAtHCID 181649—
ReactantAntipyric acidHCID 246564—
ReactantCabozantinib ImpurityHCID 136350300—
SolventWaterHCID 962—
SolventDimethylformamideHCID 6228—
ProductN-(4-((7-hydroxy-6-methoxyquinolin-4-yl)oxy)phenyl)-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamideHCID 13635030193.6%

Reaction Conditions

Temperature60 °C

Reaction Steps

To a solution of 4-(4-aminophenoxy)-6-methoxyquinolin-7-ol (3.61 g, 12.8 mmol) and 1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxylic acid (2.85 g, 12.27 mmol) in DMF (50 mL) was added EDCI (2.81 g, 14.66 mmol) and HOAT (0.33 g, 2.4 mmol). The reaction was stirred at 60° C. for 10 hours, cooled to room temperature and diluted with H2O (200 mL). The solid was collected by filtration and dried in vacuo at 60° C. overnight to give the title compound as a white solid (5.7 g, 89.9%).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09133162B2
Source datasetuspto-grants-2015_09
ORD IDord-0c68dcc7436349f6bb0aca6e57a8baea
Source noteuspto-grants-2015_09