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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 2279105Generated: November 1, 2026

4-Benzyloxy-phenylboronic acid → 6-(4-Benzyloxy-phenyl)-3-methyl-1-(tetrahydro-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid

https://huagongshe.com/reaction/2279105

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-Benzyloxy-phenylboronic acidHCID 2734314—
Reactant6-bromo-3-methyl-1-(tetrahydro-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid ethyl esterHCID 86680319—
Product6-(4-Benzyloxy-phenyl)-3-methyl-1-(tetrahydro-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acidHCID 90013694—

Reaction Steps

In analogy to Example 1 step (c) the title compound was synthesized starting from 6-bromo-3-methyl-1-(tetrahydro-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid ethyl ester and 4-benzyloxy-phenylboronic acid.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09133181B2
Source datasetuspto-grants-2015_09
ORD IDord-41b9d20e23a0479d8c312ff9ca7e4f3a
Source noteuspto-grants-2015_09