(1S,2R)-Cyclohexane-1,2-diamine, N1-BOC protected → HCID 89484469, compound

Participants

Reaction Steps

In accordance with Example 3 (Steps 1 to 4), 1-isopropyl-1H-indol-4-amine obtained in Example 45 was used instead of 1-methyl-1H-indol-4-amine, and tert-butyl((2R,3R)-3-amino-1-methoxybutan-2-yl)carbamate obtained in the above-described Step 1 was used instead of tert-butyl((1S,2R)-2-aminocyclohexyl)carbamate to obtain the titled compound as a light yellow solid.

Provenance & Evidence