(2-Aminophenyl)boronic acid → HCID 59924791, compound

HRID 2300864Notes

Reaction equation

HRID 2300864 reaction equation
[C:1]1([C@@H:7]([NH:9][C:10]2[N:15]=[C:14]([N:16]3[C:20]4[CH:21]=[CH:22][C:23](I)=[CH:24][C:19]=4[N:18]=[CH:17]3)[CH:13]=[CH:12][N:11]=2)[CH3:8])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.[NH2:26][C:27]1[CH:32]=[CH:31][CH:30]=[CH:29][C:28]=1B(O)O>>[C:1]1([C@@H:7]([NH:9][C:10]2[N:15]=[C:14]([N:16]3[C:20]4[CH:21]=[CH:22][C:23]([C:28]5[CH:29]=[CH:30][CH:31]=[CH:32][C:27]=5[NH2:26])=[CH:24][C:19]=4[N:18]=[CH:17]3)[CH:13]=[CH:12][N:11]=2)[CH3:8])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1

Participants

3

Reactant 2

HCID 2773216(2-Aminophenyl)boronic acidHCID 59924653HCID 59924653, compound

Product 1

HCID 59924791HCID 59924791, compound

Procedure

The title compound was prepared according to the procedure described in EXAMPLE 397, starting from 2-[(S)-1-Phenylethylamino]-4-[5-iodobenzimidazol-1-yl]pyrimidine and 2-aminophenylboronic acid. Mass spectrum (ESI) 437.3 (M+1).

Sources & evidence

ORD record
ord-cbeea9d5eee54ca39d16f7e5ec086ef7
Source dataset
uspto-grants-2002_12
Patent number
US06498165B1

Reaction notes

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