Pyridine, 4-bromo-2,3,5,6-tetrafluoro- → HCID 59924881, compound

HRID 2300877Notes

Reaction equation

HRID 2300877 reaction equation
[C:1]1([C@@H:7]([NH:9][C:10]2[N:15]=[C:14]([N:16]3[C:20]4[CH:21]=[CH:22][C:23]([Sn](C)(C)C)=[CH:24][C:19]=4[N:18]=[CH:17]3)[CH:13]=[CH:12][N:11]=2)[CH3:8])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.Br[C:30]1[C:35]([F:36])=[C:34]([F:37])[N:33]=[C:32]([F:38])[C:31]=1[F:39]>>[C:1]1([C@@H:7]([NH:9][C:10]2[N:15]=[C:14]([N:16]3[C:20]4[CH:21]=[CH:22][C:23]([C:30]5[C:35]([F:36])=[C:34]([F:37])[N:33]=[C:32]([F:38])[C:31]=5[F:39])=[CH:24][C:19]=4[N:18]=[CH:17]3)[CH:13]=[CH:12][N:11]=2)[CH3:8])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1

Participants

3

Reactant 2

HCID 137965Pyridine, 4-bromo-2,3,5,6-tetrafluoro-HCID 69963704HCID 69963704, compound

Product 1

HCID 59924881HCID 59924881, compound

Procedure

The title compound was prepared according to the procedure described in EXAMPLE 424, starting from 2-[(S)-1-Phenylethylamino]-4-[5-trimethylstannylbenzimidazol-1-yl]pyrimidine and 4-bromo-2,3,5,6-tetrafluoropyridine. Mass spectrum (ESI) 465.5 (M+1).

Sources & evidence

ORD record
ord-e3894c4d90774da898ac6077ed7d900a
Source dataset
uspto-grants-2002_12
Patent number
US06498165B1

Reaction notes

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