Benzo[b]furan-2-boronic acid → HCID 18373369, compound
Reaction equation
Br[C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[N:7]([CH2:11][C:12]1[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=1)[CH:6]=[C:5]2[CH2:18][C:19]([OH:21])=[O:20].[O:22]1[C:26](B(O)O)=[CH:25][C:24]2[CH:30]=[CH:31][CH:32]=[CH:33][C:23]1=2>>[O:22]1[C:23]2[CH:33]=[CH:32][CH:31]=[CH:30][C:24]=2[CH:25]=[C:26]1[C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[N:7]([CH2:11][C:12]1[CH:17]=[CH:16][CH:15]=[CH:14][CH:13]=1)[CH:6]=[C:5]2[CH2:18][C:19]([OH:21])=[O:20]Participants
3
Procedure
The title compound was prepared according to the procedure described in Example 78 except that 2-[5-bromo-1-benzyl-1H-indol-3-yl]acetic acid and benzo[b]furan-2-boronic acid were used.
Sources & evidence
- ORD record
- ord-1135265fa1dc4c61a38495723aa562eb
- Source dataset
- uspto-grants-2002_12
- Patent number
- US06500853B1
Reaction notes
Loading…