HCID 178499385, compound → HCID 178513010, compound

HRID 2301991Notes

Reaction equation

HRID 2301991 reaction equation
FC(F)(F)C(O)=O.COC(=O)CC1CC2C(=CC(OCCCCNC(N)=N)=CC=2)NC1=O.C[O:34][C:35](=[O:62])[CH2:36][C:37]1[C:38](=[O:61])[N:39]([CH2:54][C:55]2[CH:60]=[CH:59][CH:58]=[CH:57][CH:56]=2)[C:40]2[C:45]([CH:46]=1)=[CH:44][CH:43]=[C:42]([O:47][CH2:48][CH2:49][NH:50][C:51]([NH2:53])=[NH:52])[CH:41]=2>>[CH2:54]([N:39]1[C:40]2[C:45](=[CH:44][CH:43]=[C:42]([O:47][CH2:48][CH2:49][NH:50][C:51]([NH2:53])=[NH:52])[CH:41]=2)[CH:46]=[C:37]([CH2:36][C:35]([OH:62])=[O:34])[C:38]1=[O:61])[C:55]1[CH:60]=[CH:59][CH:58]=[CH:57][CH:56]=1

Participants

3

Reactant 2

HCID 178499385HCID 178499385, compoundHCID 178499393HCID 178499393, compound

Product 1

HCID 178513010HCID 178513010, compound

Procedure

The title compound is prepared according to the procedure of Example 84 except that [7-(4-guanidino-butoxy)-2-oxo-1,2,3,4-tetrahydro-quinolin-3-yl]acetic acid methyl ester trifluoroacetate is replaced with [1-benzyl-7-(2-guanidino-ethoxy)-2-oxo-1,2-dihydro-quinolin-3-yl]acetic acid methyl ester.

Sources & evidence

ORD record
ord-2af97857b74a4116978b83a6f35baa8f
Source dataset
uspto-grants-2002_08
Patent number
US06429214B1

Reaction notes

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