4-Methoxy-7-morpholinobenzo[d]thiazol-2-amine → HCID 10116462, compound

HRID 2308521Notes

Reaction equation

HRID 2308521 reaction equation
[NH2:1][C:2]1[S:3][C:4]2[C:10]([N:11]3[CH2:16][CH2:15][O:14][CH2:13][CH2:12]3)=[CH:9][CH:8]=[C:7]([O:17][CH3:18])[C:5]=2[N:6]=1.[C:19]([O:23][C:24]([N:26]1[CH2:31][CH2:30][CH:29]([C:32](Cl)=[O:33])[CH2:28][CH2:27]1)=[O:25])([CH3:22])([CH3:21])[CH3:20]>>[C:19]([O:23][C:24]([N:26]1[CH2:31][CH2:30][CH:29]([C:32](=[O:33])[NH:1][C:2]2[S:3][C:4]3[C:10]([N:11]4[CH2:16][CH2:15][O:14][CH2:13][CH2:12]4)=[CH:9][CH:8]=[C:7]([O:17][CH3:18])[C:5]=3[N:6]=2)[CH2:28][CH2:27]1)=[O:25])([CH3:22])([CH3:21])[CH3:20]

Participants

3

Reactant 2

HCID 114028614-Methoxy-7-morpholinobenzo[d]thiazol-2-amineHCID 21906247HCID 21906247, compound

Product 1

HCID 10116462HCID 10116462, compound

Procedure

Using 2-amino-4-methoxy-7-morpholin-4-yl-benzothiazol and 4-chlorocarbonyl-piperidine-1-carboxylic acid tert-butyl ester the title compound was obtained as a white solid (3%), MS: m/e=477(M+H+).

Sources & evidence

ORD record
ord-d16e83e298ef42e0809055a0ef5e786d
Source dataset
uspto-grants-2004_12
Patent number
US06835732B2

Reaction notes

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