Indole-5-carboxaldehyde → HCID 86612423, compound

HRID 2355241Notes

Reaction equation

HRID 2355241 reaction equation
[NH:1]1[C:9]2[C:4](=[CH:5][C:6]([CH:10]=[O:11])=[CH:7][CH:8]=2)[CH:3]=[CH:2]1.[C:12]([O:16][C:17]([N:19]1[C:24]([CH3:26])([CH3:25])[CH2:23][CH2:22]OS1(=O)=O)=[O:18])([CH3:15])([CH3:14])[CH3:13]>>[C:12]([O:16][C:17]([NH:19][C:24]([CH3:25])([CH3:26])[CH2:23][CH2:22][N:1]1[C:9]2[C:4](=[CH:5][C:6]([CH:10]=[O:11])=[CH:7][CH:8]=2)[CH:3]=[CH:2]1)=[O:18])([CH3:15])([CH3:14])[CH3:13]

Participants

3

Reactant 2

HCID 589040Indole-5-carboxaldehydeHCID 59383129HCID 59383129, compound

Product 1

HCID 86612423HCID 86612423, compound

Procedure

Prepared analogously to Component V(a) by alkylation of indole-5-carbaldehyde with N-tert-butoxycarbonyl-4,4-dimethyl-[1,2,3]oxathiazinane-2,2-dioxide (Component XI).

Sources & evidence

ORD record
ord-ab776c10f0124b30a8f476f7559ad14c
Source dataset
uspto-grants-2010_07
Patent number
US07754756B2

Reaction notes

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