Carbamate → HCID 11362125, compound

HRID 2358295Notes

Reaction equation

[NH2:1][CH:2](C1C2CCCCC=2C=CC=1)[CH2:3][N:4]1[C:13]([C:14]#[N:15])=[C:12]([C:16]2[CH:21]=[CH:20][CH:19]=[CH:18][CH:17]=2)[C:11]2[C:6](=[CH:7][CH:8]=[C:9]([O:22][CH3:23])[CH:10]=2)[C:5]1=[O:24].[C:35](=[O:38])([O-:37])N>>[C:6]([O:37][C:35](=[O:38])[NH:1][CH2:2][CH2:3][N:4]1[C:13]([C:14]#[N:15])=[C:12]([C:16]2[CH:21]=[CH:20][CH:19]=[CH:18][CH:17]=2)[C:11]2[C:6](=[CH:7][CH:8]=[C:9]([O:22][CH3:23])[CH:10]=2)[C:5]1=[O:24])([CH3:11])([CH3:7])[CH3:5]

Participants

Reactant 2

HCID 276Carbamate

HCID 68717879HCID 68717879, compound

Product 1

HCID 11362125HCID 11362125, compound

Procedure

Compound 56a was prepared essentially according to the procedure described above in Example I for compound 8 by using tert-butyl-N-2-aminoethyl)-carbamate in place of aminoacetaldehyde diethyl acetal in Step D.

Sources & evidence

ORD record: ord-a421ddd702f14649ad5cf224422898fa
Source dataset: uspto-grants-2010_07
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US07763614B2

Reaction notes

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