2-Bromopyrimidine → [4-(Pyrimidin-2-yl)phenyl]methanol

Participants

Reaction Steps

Reaction and post-treatment were carried out in the same manlier as in Reference Example 13 except for using 4-hydroxymethylphenylboronic acid (144 mg, 0.948 mmol), and using 2-bromopyrimidine (101 mg, 0.635 mmol) in place of 4-bromopyridazine to afford the title compound (119 mg) substantially quantitatively as a slightly yellow solid.

Provenance & Evidence