3-Fluorobenzoyl chloride → HCID 58711984, compound

Participants

Reaction Steps

In a similar manner as described for Intermediate 59, using 6-(1-aminoethyl)-N-[4-(methyloxy)phenyl]-1,2,4-triazin-3-amine (Intermediate 47) (100 mg, 0.41 mmol), and 3-fluorobenzoyl chloride (0.059 mL, 0.45 mmol) to afford 3-fluoro-N-[1-(3-{[4-(methyloxy)phenyl]amino}-1,2,4-triazin-6-yl)ethyl]benzamide (130 mg) as a yellow solid. MS m/z 368 (M+1).

Provenance & Evidence