2-Bromo-4-fluoro-1-(methoxymethoxymethyl)benzene → HCID 11299354, compound

HRID 2375779Notes

Reaction equation

HRID 2375779 reaction equation
[C:1]([C:3]1[CH:4]=[C:5]([B:9]2[O:13][CH2:12][CH2:11]O2)[CH:6]=[CH:7][CH:8]=1)#[N:2].Br[C:15]1[CH:20]=[C:19]([F:21])[CH:18]=[CH:17]C=1COCOC>>[F:21][C:19]1[CH:18]=[CH:17][C:11]2[CH2:12][O:13][B:9]([C:5]3[CH:4]=[C:3]([CH:8]=[CH:7][CH:6]=3)[C:1]#[N:2])[C:15]=2[CH:20]=1

Participants

3

Reactant 2

HCID 667046952-Bromo-4-fluoro-1-(methoxymethoxymethyl)benzeneHCID 667383483-(1,3,2-Dioxaborolan-2-yl)benzonitrile

Product 1

HCID 11299354HCID 11299354, compound

Procedure

This was prepared as per the procedure in Example 11, from 2-(3-cyanophenyl)-[1,3,2]-dioxaborolane and 1-bromo-5-fluoro-2-((methoxymethoxy)methyl)benzene to afford white crystalline product.

Workup

  1. customto afford white crystalline product

Sources & evidence

ORD record
ord-e02703cdea224375bbb6713344483143
Source dataset
uspto-grants-2008_12
Patent number
US07465836B2

Reaction notes

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