4-Fluorophenylboronic acid → HCID 59442947, compound

HRID 2380906Notes

Reaction equation

HRID 2380906 reaction equation
FC(F)(F)S(O[C:7]1[C:16]2[C:11](=[CH:12][C:13]([O:17][Si](C(C)(C)C)(C)C)=[CH:14][CH:15]=2)[O:10][C:9]([CH3:26])([CH3:25])[CH:8]=1)(=O)=O.[F:29][C:30]1[CH:35]=[CH:34][C:33](B(O)O)=[CH:32][CH:31]=1>>[F:29][C:30]1[CH:35]=[CH:34][C:33]([C:7]2[C:16]3[C:11](=[CH:12][C:13]([OH:17])=[CH:14][CH:15]=3)[O:10][C:9]([CH3:25])([CH3:26])[CH:8]=2)=[CH:32][CH:31]=1

Participants

3

Reactant 2

HCID 2856454-Fluorophenylboronic acidHCID 59442939HCID 59442939, compound

Product 1

HCID 59442947HCID 59442947, compound

Procedure

The compound obtained in (1) described above (8 g) and 4-fluorophenylboronic acid (3.07 g) were treated in the same manner as Reference Example 37(4) to give the titled compound (4.6 g) as a colorless powder.

Sources & evidence

ORD record
ord-b0d5267798c2474a8bec43557d92170d
Source dataset
uspto-grants-2012_09
Patent number
US08258131B2

Reaction notes

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