3-Methanesulfonylbenzoic acid → N-[5-(3-furyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-3-(methylsulfonyl)benzamide

Participants

Reaction Steps

The title compound was prepared following procedure described for example 2, but starting from 5-(3-furyl)[1,2,4]triazolo[1,5-a]pyridin-2-amine ((A2), 50 mg; 0.25 mmol; 1.0 eq.) and 3-methylsulphonylbenzoic acid (60 mg, 0.3 mmol, 1.2 eq.) as an off-white solid (9 mg, 9%). HPLC, Rt: 2.79 min. (purity 96.5%). LC/MS, M+(ESI): 383.0, M−(ESI): 381.0.

Provenance & Evidence