(R)-8-(benzyloxy)-5-(2-bromo-1-((tert-butyldimethylsilyl)oxy)ethyl)quinolin-2(1H)-one → HCID 59145945, compound

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The title compound was prepared from (R)-({-[(1-{2-[4-(2-aminoethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-1,2,4-triazol-3-yl}(cyclohexyl)phenylmethanol (Preparation 13, 2.57 g, 5.12 mmol) and 8-(benzyloxy)-5-[(1R)-2-bromo-1-{[tert-butyl(dimethyl)silyl]oxy}ethyl]quinolin-2(1H)-one (WO2005/09286, 2.50 g, 5.12 mmol) using the same method as described in preparation 7 to give a white solid, in 40% yield, 2.3 g.

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