4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzoic Acid → HCID 9870601, compound

HRID 2392687Notes

Reaction equation

HRID 2392687 reaction equation
[CH3:1][C:2]1[CH:7]=[C:6]([C:8]2[N:12]=[C:11]([CH3:13])[O:10][N:9]=2)[CH:5]=[CH:4][C:3]=1[C:14]1[CH:19]=[CH:18][C:17]([C:20]([OH:22])=O)=[CH:16][CH:15]=1.[CH3:23][N:24]([CH3:38])[CH2:25][CH2:26][CH2:27][O:28][C:29]1[CH:30]=[C:31]([CH:33]=[CH:34][C:35]=1[O:36][CH3:37])[NH2:32]>>[CH3:38][N:24]([CH3:23])[CH2:25][CH2:26][CH2:27][O:28][C:29]1[CH:30]=[C:31]([NH:32][C:20]([C:17]2[CH:18]=[CH:19][C:14]([C:3]3[CH:4]=[CH:5][C:6]([C:8]4[N:12]=[C:11]([CH3:13])[O:10][N:9]=4)=[CH:7][C:2]=3[CH3:1])=[CH:15][CH:16]=2)=[O:22])[CH:33]=[CH:34][C:35]=1[O:36][CH3:37]

Participants

3

Reactant 2

HCID 111301684-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzoic AcidHCID 18980073HCID 18980073, compound

Product 1

HCID 9870601HCID 9870601, compound

Procedure

The title compound was prepared from 2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)biphenyl-4-carboxylic acid (EP 0533268 A1) and 3-(3-dimethylaminopropoxy)-4-methoxyaniline (D23) using a similar procedure to Example 1 (58%).

Sources & evidence

ORD record
ord-84fe6ade32d74a00beac918b5b8f546a
Source dataset
uspto-grants-1998_09
Patent number
US05801170

Reaction notes

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