HuagongsheHuagongshe Chemistry Print Report · For research reference only
HCID 43665761, compound → HCID 71252517, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | HCID 43665761 | HCID 43665761 | — |
| Reactant | 1-(5-Cyclopropyl-3-methylpyridin-2-yl)piperazine | HCID 58484718 | — |
| Product | HCID 71252517 | HCID 71252517 | 70.6% |
Reaction Steps
Using 4-[2-(1,1-dioxo-1λ6-isothiazolidin-2-yl)ethyl]benzoic acid (162 mg) described in Preparation Example 41 and 1-(5-cyclopropyl-3-methylpyridin-2-yl)piperazine (130 mg) described in Preparation Example 83 and by the reaction and treatment in the same manner as in Example 87, the title compound (198 mg) was obtained.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08816079B2 |
| Source dataset | uspto-grants-2014_08 |
| ORD ID | ord-e4f11c98170a49bfb11c12a18b3ea3d5 |
| Source note | uspto-grants-2014_08 |