HuagongsheHuagongshe Chemistry Print Report · For research reference only
1,3-Propanesultam → HCID 71252205, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1,3-Propanesultam | HCID 642157 | — |
| Reactant | HCID 71252060 | HCID 71252060 | — |
| Product | HCID 71252205 | HCID 71252205 | 52.6% |
Reaction Steps
Using 1-acetyl-3-{5-chloro-2-[4-(3,5,6-trimethylpyridin-2-yl)piperazine-1-carbonyl]phenyl}imidazolidin-2-one (190 mg) described in Preparation Example 258 and isothiazolidine 1,1-dioxide (73 mg) and by the reaction and treatment in the same manner as in Example 649, the title compound (109 mg) was obtained.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08816079B2 |
| Source dataset | uspto-grants-2014_08 |
| ORD ID | ord-00986de1dddf4a3ca068317700e5e8d7 |
| Source note | uspto-grants-2014_08 |