Benzyl Alcohol → HCID 178420404, compound

HRID 2420580Notes

Reaction equation

HRID 2420580 reaction equation
[CH3:1][O:2][C:3]1[C:8]2[CH:9]=[N:10][C:11]3[NH:15][N:14]=[CH:13][C:12]=3[C:7]=2[N:6]2[N:16]=[CH:17][N:18]=[C:5]2[N:4]=1.ClC1C2C=NC3N(CC)N=CC=3C=2N2N=CN=C2N=1.C(O)[C:39]1[CH:44]=[CH:43][CH:42]=[CH:41][CH:40]=1>C(O)C>[C:39]1([CH2:1][O:2][C:3]2[C:8]3[CH:9]=[N:10][C:11]4[NH:15][N:14]=[CH:13][C:12]=4[C:7]=3[N:6]3[N:16]=[CH:17][N:18]=[C:5]3[N:4]=2)[CH:44]=[CH:43][CH:42]=[CH:41][CH:40]=1

Participants

5

Reactant 3

HCID 244Benzyl AlcoholHCID 227584865-Chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]-triazolo[1,5-a]pyrimidineHCID 178494003HCID 178494003, compound

Product 1

HCID 178420404HCID 178420404, compound

Reagents, catalysts & solvents 1

HCID 702EthanolSolvent

Procedure

By substituting the 5-chloro-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine of Example 15 for the 5-chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine and benzyl alcohol for the ethanol in the procedure of Example 4, 5-phenylmethoxy-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine is obtained.

Sources & evidence

ORD record
ord-aee5f1c3ef804bb8a316538257da55c0
Source dataset
uspto-grants-1978_08
Patent number
US04110454

Reaction notes

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