HuagongsheHuagongshe Chemistry Print Report · For research reference only
Anthranilic Acid → 3-Methyl-2-[2-methyl-4-(1-cyclopentyl-4-piperidinyloxy)-phenyl]-4(3H)-quinazolinone
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Anthranilic Acid | HCID 227 | — |
| Reactant | Methylamine | HCID 6329 | — |
| Reactant | Cyclopentanone | HCID 8452 | — |
| Reactant | 4-Methoxy-2-methylbenzaldehyde | HCID 283285 | — |
| Reactant | Tert-butyl 4-hydroxypiperidine-1-carboxylate | HCID 643502 | — |
| Product | 3-Methyl-2-[2-methyl-4-(1-cyclopentyl-4-piperidinyloxy)-phenyl]-4(3H)-quinazolinone | HCID 11690234 | — |
Reaction Steps
The entitled compound was obtained according to the method of Example 85 but using anthranilic acid, methylamine, 2-methyl-4-methoxybenzaldehyde, tert-butyl 4-hydroxytetrahydro-1(2H)-pyridinecarboxylate, and cyclopentanone.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07960394B2 |
| Source dataset | uspto-grants-2011_06 |
| ORD ID | ord-c0c3cfacf65140b7b5fe8b871bb6df5a |
| Source note | uspto-grants-2011_06 |