HuagongsheHuagongshe Chemistry Print Report · For research reference only
Allyl 2,2,2-Trichloroacetimidate → benzyloxycarbonyl-beta-(allylamino)-L-alanine, methyl ester
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Allyl 2,2,2-Trichloroacetimidate | HCID 316905 | — |
| Reactant | 3-Amino-N-((phenylmethoxy)carbonyl)-L-alanine methyl ester | HCID 11043221 | — |
| Product | benzyloxycarbonyl-beta-(allylamino)-L-alanine, methyl ester | HCID 131719024 | — |
Reaction Steps
The β-amino functionality of Nα -(benzyloxycarbonyl)-β-(amino)-L-alanine, methyl ester is then allylated with allyl trichloroacetimidate to give the corresponding Nα -(benzyloxycarbonyl)-β-(allylamino)-L-alanine, methyl ester using conditions described previously in Scheme F, step b.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US05527795 |
| Source dataset | uspto-grants-1996_06 |
| ORD ID | ord-294c398671904d6d8a7309e44f113570 |
| Source note | uspto-grants-1996_06 |