Formamide, N-1-naphthalenyl- → 1-[N-(1-Azabicyclo[3.3.0]octan-5-yl)methyl-N-formylamino]-naphthalene

Participants

Reaction Steps

The procedures described in Example 2 were repeated except that N-formyl-1-naphthylamine (1.83 g, 10.7 mmol ) and 5-chloromethyl-1-azabicyclo[3.3.0]octane (hydrochloride, 2.30 g, 11.7 mmol) were employed. In this case, the desired compound was obtained as a colorless liquid (3.02 g, 95.9%

Provenance & Evidence