HCID 12218835, compound → HCID 12593080, compound

HRID 261085Notes

Reaction equation

HRID 261085 reaction equation
[C:1]([CH2:4][C:5]1[CH:13]=[CH:12][C:11]([NH:14][CH3:15])=[CH:10][C:6]=1[C:7]([OH:9])=O)(O)=O.Br.[NH2:17][CH2:18][CH2:19][CH2:20][SH:21]>>[CH3:15][NH:14][C:11]1[CH:12]=[CH:13][C:5]2[CH:4]=[C:1]3[S:21][CH2:20][CH2:19][CH2:18][N:17]3[C:7](=[O:9])[C:6]=2[CH:10]=1

Participants

3

Reactant 2

HCID 12218835HCID 12218835, compoundHCID 12593127HCID 12593127, compound

Product 1

HCID 12593080HCID 12593080, compound

Procedure

By following the same procedure as in Example 29 using 2.3 g. of 2-carboxymethyl-5-methylaminobenzoic acid and 1.8 g. of 3-aminopropanethiol.hydrobromide, 300 mg. of 8-methylamino-6-oxo-3,4-dihydro-2H,6H-1,3-thiazino[3,2-b]isoquinoline was obtained.

Sources & evidence

ORD record
ord-cd36e8f5e7d24d56b82b858472969e14
Source dataset
uspto-grants-1979_08
Patent number
US04163844

Reaction notes

Loading…