Sodium borohydride → HCID 57141280, compound

Participants

Reaction Steps

155 mg (0.266 mmol) of (2R*,4S*)-2-benzyl-1-(2-quinolinylcarbonyl)-N-(4-quinolylmethyl)-N-trifluoroacetyl-4-piperidinamine are reacted with 40 mg (1.06 mmol) of sodium borohydride in analogy to Example 2. The title compound ##STR34## is obtained as white foam. TLC: methylene chloride/methanol/conc. ammonia (700:50:1) Rf =0.42, D-MS: M+ =486.

Provenance & Evidence