反应详情

80 mg (0.142 mmol) of (2R*,4S*)-2-benzyl-1-(benzyloxycarbonyl)-N-(4-quinolylmethyl)-N-trifluoroacetyl-4-piperidinamine are reacted with 22 mg (0.57 mmol) of sodium borohydride in analogy to Example 2. The title compound ##STR36## is obtained as colourless oil. TLC: methylene chloride/methanol/conc. ammonia (700:50:1) Rf =0.43, FD-MS: M+ =465.