Sodium borohydride → HCID 57042465, compound

Participants

Reaction Steps

230 mg (0.409 mmol) of (2R*,4S*)-2-benzyl-1-(3-methoxybenzoyl)-N-(4-quinolylmethyl)-N-trifluoroacetyl-4-piperidinamine are reacted with 81 mg (2.14 mmol) of sodium borohydride in analogy to Example 2. The title compound of the formula ##STR48## is obtained as white foam. TLC: methylene chloride/methanol/conc. ammonia (1000:50:1) Rf =0.26, FD-MS: M+ =465.

Provenance & Evidence