HuagongsheHuagongshe Chemistry Print Report · For research reference only
1-Tosyl-1H-pyrrolo(2,3-B)pyridine-4-boronic acid pinacol ester → 4-[2-methyl-4-(4-nitrophenyl)-1,3-thiazol-5-yl]-1-[(4-methylphenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1-Tosyl-1H-pyrrolo(2,3-B)pyridine-4-boronic acid pinacol ester | HCID 49758926 | — |
| Reactant | 5-Bromo-2-methyl-4-(4-nitrophenyl)-1,3-thiazole | HCID 68998100 | — |
| Product | 4-[2-methyl-4-(4-nitrophenyl)-1,3-thiazol-5-yl]-1-[(4-methylphenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine | HCID 69001198 | — |
Reaction Steps
Following the procedure described for Intermediate 6 with 5-bromo-2-methyl-4-(4-nitrophenyl)-1,3-thiazole and [(4-methylphenyl)sulfonyl]-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrrolo[2,3-b]pyridine provided title compound. ESMS [M+H]+: 491.2
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07419988B2 |
| Source dataset | uspto-grants-2008_09 |
| ORD ID | ord-dd0dd00fd49d4c54a924b1c45fed940e |
| Source note | uspto-grants-2008_09 |