1-(Phenylsulfonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-pyrrolo[2,3-B]pyridine-2-carboxaldehyde → N-(4-{4-[2-formyl-1-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethyl-1H-pyrazol-3-yl}phenyl)-N'-phenylurea

Participants

Role	Name	HCID	Charge
Reactant	1-(Phenylsulfonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-pyrrolo[2,3-B]pyridine-2-carboxaldehyde	HCID 46236899	—
Reactant	N-[4-(4-Bromo-1-ethyl-1H-pyrazol-3-yl)phenyl]-N′-phenylurea	HCID 68997560	—
Product	N-(4-{4-[2-formyl-1-(phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-ethyl-1H-pyrazol-3-yl}phenyl)-N'-phenylurea	HCID 46236618	—

Reaction Steps

Following the procedure described in Intermediate 100 with N-[4-(4-bromo-1-ethyl-1H-pyrazol-3-yl)phenyl]-N′-phenylurea and 1-(phenylsulfonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrrolo[2,3-b]pyridine-2-carbaldehyde provided the title compound. ESMS [M+H]+: 591.4

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US07419988B2
Source dataset	uspto-grants-2008_09
ORD ID	ord-53b034e6f51a439b97d79b6d3513d28e
Source note	uspto-grants-2008_09