HCID 22008823, compound → HCID 20641951, compound

HRID 322003Notes

Reaction equation

HRID 322003 reaction equation
[ClH:1].Cl.[NH2:3][C:4]1[CH:12]=[CH:11][CH:10]=[C:9]([F:13])[C:5]=1[C:6]([NH2:8])=[NH:7].Cl[C:15]1[C:23](Cl)=[CH:22][CH:21]=[C:20]2[C:16]=1[C:17](=[O:30])[N:18]1[CH2:28][CH2:27][C:26](=O)[CH2:25][CH:19]12>>[NH2:7][C:6]1[C:5]2[C:4](=[CH:12][CH:11]=[CH:10][C:9]=2[F:13])[NH:3][C:26]2([CH2:27][CH2:28][N:18]3[C:17](=[O:30])[C:16]4[C:20]([CH:19]3[CH2:25]2)=[C:21]([Cl:1])[CH:22]=[CH:23][CH:15]=4)[N:8]=1

Participants

3

Reactant 2

HCID 22008823HCID 22008823, compoundHCID 22008829HCID 22008829, compound

Product 1

HCID 20641951HCID 20641951, compound

Procedure

The compounds of Examples 15 and 16 were prepared from 2-amino-6-fluorobenzamidine dihydrochloride and 7,8-dichloro-1,3,4,10b-tetrahydropyrido[2,1-a]isoindole-2,6-dione (Preparation 5).

Sources & evidence

ORD record
ord-ec4b7a4ea27a457b8f8b7603b20b9f10
Source dataset
uspto-grants-2001_04
Patent number
US06211189B1

Reaction notes

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