3-Fluoro-4-methylbenzeneboronic acid → 2-(3-Fluoro-4-methylphenyl)-5-Methoxy-3-phenyl-1H-inden-1-one

Participants

Reaction Steps

The procedure of Step 7 of Example 1 was repeated except for using 2-bromo-5-methoxy-3-phenyl-1H-inden-1-one obtained in Step 4 of Example 129 as a starting material instead of 6-(2-morpholinoethoxy)-2-bromo-3-phenyl-1H-inden-1-one, 3-fluoro-4-methylphenylboronic acid instead of 3-pyridinylboronic acid, and being stirred for 10 min to obtain the title compound (65%).

Provenance & Evidence