反应详情

The title compound, white solid (31 mg, 31%), MS (ISP) m/z=401.5 [(M+H)+], mp 158° C., was prepared in accordance with the general method of example 1 from trans-4-{2-[4-(2,3-dihydro-benzofuran-4-yl)-piperidin-1-yl]-ethyl}-cyclohexylamine dihydrochloride (intermediate B) (100 mg, 0.25 mmol) and 3-hydroxy-propionic acid.