Benzenesulfonyl chloride → HCID 178527577, compound

Participants

Reaction Steps

The title compound, white solid (96 mg, 82%), MS (ISP) m/z=469.4 [(M+H)+], mp 130° C., was prepared in accordance with the general method of example 47 from trans-4-{2-[4-(2,3-dihydro-benzofuran-4-yl)-piperidin-1-yl]-ethyl}-cyclohexylamine dihydro chloride (intermediate B) (100 mg, 0.25 mmol) and benzenesulfonyl chloride.

Provenance & Evidence