Isocaproic acid → HCID 178445240, compound

Participants

Reaction Steps

The title compound, white solid (77 mg, 73%), MS (ISP) m/z=427.4 [(M+H)+], mp 188° C., was prepared in accordance with the general method of example 1 from trans-4-{2-[4-(2,3-dihydro-benzofuran-4-yl)-piperidin-1-yl]-ethyl}-cyclohexylamine dihydro chloride (intermediate B) (100 mg, 0.25 mmol) and 4-methyl-pentanoic acid.

Provenance & Evidence