Hydrochloric Acid → HCID 70197051, compound

Participants

Reaction Steps

By steps analogous to steps (a) to (c) of Synthetic Example 14, the product from step (a) was converted to (R)-3-(1-methyl-1,2,3,6-tetrahydro-4-pyridyl)-5-(2-oxo-1,3-oxazolidin-4-ylmethyl)-1H-indole hydrate, mp 229°-231° C., [α]D18 +24.9° (c=0.5, 1N aqu. HCl). Elemental analysis and 1H NMR were consistent with the proposed structure.

Provenance & Evidence