Back
HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 344343Generated: October 31, 2026

Phenyl isocyanate → HCID 57237769, compound

https://huagongshe.com/reaction/344343

Reaction equation

Participants

RoleNameHCIDCharge
ReactantPhenyl isocyanateHCID 7672—
Reactant4-Amino-5-chloro-2-methoxybenzoic acidHCID 81626—
ReactantHCID 53706155HCID 53706155—
ProductHCID 57237769HCID 57237769—

Reaction Steps

6-((3S)-3-tert-Butoxycarbonylaminomethylpyrrolidin-1-yl)hexylamine (1.00 g) as starting compound was reacted and treated in the same manner as in Example 34 using phenyl isocyanate (0.38 ml) and 4-amino-5-chloro-2-methoxybenzoic acid (0.67 g) to give 4-amino-5-chloro-2-methoxy-N-((3S)-1-(6-(3-phenylureido)hexyl)pyrrolidin-3-ylmethyl)benzamide.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS05864039
Source datasetuspto-grants-1999_01
ORD IDord-ce59d566e05442dfad05f920eaf28f46
Source noteuspto-grants-1999_01