HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
2-Thiophenecarboxaldehyde → 4-amino-5-chloro-2-methoxy-N-((1-(5-(2-thienylmethylamino)pentyl)piperidin-4-yl)methyl)benzamide
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | 2-Thiophenecarboxaldehyde | HCID 7364 | — |
| Edukt | 4-Amino-N-(1-(5-aminopentyl)piperidin-4-ylmethyl)-5-chloro-2-methoxybenzamide | HCID 54008363 | — |
| Produkt | 4-amino-5-chloro-2-methoxy-N-((1-(5-(2-thienylmethylamino)pentyl)piperidin-4-yl)methyl)benzamide | HCID 53759958 | 99,9% |
Reaktionsschritte
4-Amino-N-(1-(5-aminopentyl)piperidin-4-ylmethyl)-5-chloro-2-methoxybenzamide (2 g) as starting compound and 2-thiophenecarboxaldehyde (0.64 g) were reacted and treated in the same manner as in Example 121 to give 2.5 g of 4-amino-5-chloro-2-methoxy-N-((1-(5-(2-thienylmethylamino)pentyl)piperidin-4-yl)methyl)benzamide.
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US05864039 |
| Quelldatensatz | uspto-grants-1999_01 |
| ORD ID | ord-965edb77c7a840769e336d0940f4fb76 |
| Quellennotiz | uspto-grants-1999_01 |